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1bqi

;USE OF PAPAIN AS A MODEL FOR THE STRUCTURE-BASED DESIGN OF CATHEPSIN K INHIBITORS. CRYSTAL STRUCTURES OF TWO PAPAIN INHIBITOR COMPLEXES DEMONSTRATE BINDING TO S'-SUBSITES. ;

Method: X-RAY DIFFRACTION Dmax: 54.5 Å Quality: GOOD

SAXS Profile

SAXS profile for 1bqi

P(r) Distribution

P(r) distribution for 1bqi

1. Structure Basics

entry_id1bqi
deposition_date1998-08-16
title;USE OF PAPAIN AS A MODEL FOR THE STRUCTURE-BASED DESIGN OF CATHEPSIN K INHIBITORS. CRYSTAL STRUCTURES OF TWO PAPAIN INHIBITOR COMPLEXES DEMONSTRATE BINDING TO S'-SUBSITES. ;
keywordsHYDROLASE, SULFHYDRYL PROTEINASE, PAPAIN; HYDROLASE
methodX-RAY DIFFRACTION

Download Data

2. SAXS Parameters (CRYSOL)

rg_guinier17.59
rg_electron16.39
i010401300.00
molecular_weight23843.0 kDa
excluded_volume29784 ų
envelope_volume33307 ų
shell_volume16803 ų
envelope_diameter54.9
shell_rg22.69
envelope_rg16.67
shape_rg16.38
total_rg17.46
total_atoms1684
n_residues212
n_harmonics20
q_range— – 0.5000 −1
n_points101
shell_typedirectional
solvent_density0.3340 e/ų
contrast_shell0.0300 e/ų
crysol_version4.1.3

3. P(r) Analysis (GNOM)

dmax54.5
rg_real17.47
rg_real_error0.25
i0_real1.0400e+07
i0_real_error1.1920e+05
rg_reciprocal17.49
i0_reciprocal10400000.0000
total_estimate0.8986
solution_quality GOOD a GOOD solution
n_peaks2
r_peak_primary22.6
skewness0.150
kurtosis-0.422
angular_range— – 0.4500 −1
current_alpha0.0000
highest_alpha3019000.0000
n_real_points76
gnom_version4.1.3
quality_criteria AN1: 0.000; Oscil: 0.907; Stabil: 1.000; Sysdev: 1.000; Positv: 1.000; Valcen: 0.993; Smooth: 0.964

4. Crystallography & Experiment

5. Entities & Polymer Info (3)

6. Citations (1)

7. Files & Curves (10)