当前蛋白身份:P37231-2
重新检索
差异标签只比较当前检索结果;所有PDB和assembly原始记录仍分别保留。
相关结构差异明细
一行代表一个 PDB 条目中的一个 biological assembly;同一蛋白的多个单体会分别列出。
| PDB 条目 | Assembly / 聚集状态 | 构建体 | 突变与修饰 | 配体、离子与非聚合物 | 实验方法 | 实验环境 | 结构质量 |
|---|---|---|---|---|---|---|---|
| 7WGO X-ray structure of human PPAR gamma ligand binding domain-bezafibrate co-rystals obtained by co-crystallization 提交 2021-12-28 | Assembly 1 蛋白异源复合物 异源复合物;蛋白 × 2 PDB 声明:dimeric(2) 与蛋白数一致 |
链 A
203–477(275 aa)
|
未记录 | PEM 2-[P-[2-P-CHLOROBENZAMIDO)ETHYL]PHENOXY]-2-METHYLPROPIONIC ACID × 1 | X-RAY DIFFRACTION |
X-ray结晶条件
VAPOR DIFFUSION;293 K;0.1 M Tris (pH 8.0), 1.1 M trisodium citrate
|
分辨率 2.36 Å R-free 0.225 |
| 7WGP X-ray structure of human PPAR gamma ligand binding domain-fenofibric acid co-crystals obtained by co-crystallization 提交 2021-12-28 | Assembly 1 蛋白异源复合物 异源复合物;蛋白 × 2 PDB 声明:dimeric(2) 与蛋白数一致 |
链 A
203–477(275 aa)
|
未记录 | F5A 2-[4-(4-chlorobenzene-1-carbonyl)phenoxy]-2-methylpropanoic acid × 3 | X-RAY DIFFRACTION |
X-ray结晶条件
VAPOR DIFFUSION;293 K;0.1 M Tris (pH 8.0), 1.1 M trisodium citrate
|
分辨率 2.53 Å R-free 0.269 |
| 7WGQ X-ray structure of human PPAR gamma ligand binding domain-pemafibrate co-crystals obtained by co-crystallization 提交 2021-12-28 | Assembly 1 蛋白异源复合物 异源复合物;蛋白 × 2 PDB 声明:dimeric(2) 与蛋白数一致 |
链 A
203–477(275 aa)
|
未记录 | P7F (2~{R})-2-[3-[[1,3-benzoxazol-2-yl-[3-(4-methoxyphenoxy)propyl]amino]methyl]phenoxy]butanoic acid × 1 | X-RAY DIFFRACTION |
X-ray结晶条件
VAPOR DIFFUSION;293 K;0.1 M HEPES (pH 7.5), 1.1 M trisodium citrate
|
分辨率 2.43 Å R-free 0.252 |
| 8HUM X-ray structure of human PPAR gamma ligand binding domain-lanifibranor-SRC1 coactivator peptide co-crystals obtained by co-crystallization 提交 2022-12-24 | Assembly 1 蛋白异源复合物 异源复合物;蛋白 × 2 PDB 声明:dimeric(2) 与蛋白数一致 |
链 A
203–477(275 aa)
|
未记录 | BJB 4-[1-(1,3-benzothiazol-6-ylsulfonyl)-5-chloro-indol-2-yl]butanoic acid × 1 | X-RAY DIFFRACTION |
X-ray结晶条件
VAPOR DIFFUSION;293 K;0.1 M HEPES (pH 7.5), 1.0 M trisodium citrate
|
分辨率 2.29 Å R-free 0.250 |
| 8HUP X-ray structure of human PPAR gamma ligand binding domain-seladelpar-SRC1 coactivator peptide co-crystals obtained by co-crystallization 提交 2022-12-24 | Assembly 1 蛋白异源复合物 异源复合物;蛋白 × 2 PDB 声明:dimeric(2) 与蛋白数一致 |
链 A
203–477(275 aa)
|
未记录 | KKB Seladelpar × 1 | X-RAY DIFFRACTION |
X-ray结晶条件
VAPOR DIFFUSION;293 K;0.1 M Tris (pH 8.0), 1.1 M trisodium citrate
|
分辨率 2.36 Å R-free 0.234 |
| 9IWK X-ray structure of human PPARgamma ligand binding domain-NCoR2 corepressor peptide co-crystals obtained by co-crystallization 提交 2024-07-25 | Assembly 1 蛋白异源复合物 异源复合物;蛋白 × 2 PDB 声明:dimeric(2) 与蛋白数一致 |
链 A
203–477(275 aa)
|
未记录 | 未记录非水小分子 | X-RAY DIFFRACTION |
X-ray结晶条件
VAPOR DIFFUSION;293 K;0.1M Tris (pH 8.5), 30% PEG 8000, 0.2M ammonium sulfate
|
分辨率 2.43 Å R-free 0.266 |
| 9IWK X-ray structure of human PPARgamma ligand binding domain-NCoR2 corepressor peptide co-crystals obtained by co-crystallization 提交 2024-07-25 | Assembly 2 蛋白异源复合物 异源复合物;蛋白 × 2 PDB 声明:dimeric(2) 与蛋白数一致 |
链 C
203–477(275 aa)
|
未记录 | 未记录非水小分子 | X-RAY DIFFRACTION |
X-ray结晶条件
VAPOR DIFFUSION;293 K;0.1M Tris (pH 8.5), 30% PEG 8000, 0.2M ammonium sulfate
|
分辨率 2.43 Å R-free 0.266 |