1he8

Ras G12V - PI 3-kinase gamma complex

Method: X-RAY DIFFRACTION Dmax: 120.7 Å Quality: GOOD

SAXS 散射曲线 SAXS Profile

SAXS profile for 1he8

P(r) 距离分布 P(r) Distribution

P(r) distribution for 1he8
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1. 结构基本信息 1. Structure Basics

条目编号 entry_id1he8
沉积日期 deposition_date2000-11-20
结构标题 titleRas G12V - PI 3-kinase gamma complex
关键词 keywords;KINASE/HYDROLASE, COMPLEX (PHOSPHOINOSITIDE KINASE-RAS), PHOSPHOINOSITIDE 3-KINASE GAMMA - H-RAS G12V COMPLEX, PHOSPHATIDYLINOSITOL 3-KINASE, PI3K, PI 3-K, PI 3-KINASE, SECOND MESSENGER GENERATION, RAS EFFECTOR, H-RAS G12V, ONCOGENE PROTEIN, GMPPNP, GTP, RAS-BINDING DOMAIN, HEAT DOMAIN, KINASE-HYDROLASE complex ;; KINASE/HYDROLASE
实验方法 methodX-RAY DIFFRACTION

2. SAXS 参数 (CRYSOL 理论计算) 2. SAXS Parameters (CRYSOL)

回转半径 Rg (Guinier) rg_guinier33.98
回转半径 Rg (电子) rg_electron33.49
零角强度 I(0) i0169990000.00
分子量 molecular_weight105690.0 kDa
排除体积 excluded_volume132910 ų
包络体积 envelope_volume167980 ų
水化壳体积 shell_volume43687 ų
包络直径 envelope_diameter127.7
壳层 Rg shell_rg38.45
包络 Rg envelope_rg33.35
形状 Rg shape_rg33.49
总 Rg total_rg33.88
总原子数 total_atoms7428
残基数 n_residues915
球谐函数阶数 n_harmonics20
q 范围 q_range— – 0.5000 −1
数据点数 n_points101
壳层类型 shell_typedirectional
溶剂电子密度 solvent_density0.3340 e/ų
壳层衬度 contrast_shell0.0300 e/ų
CRYSOL 版本 crysol_version4.1.3

3. P(r) 距离分布 (GNOM 反演) 3. P(r) Analysis (GNOM)

最大尺寸 Dmax dmax120.7
Rg (实空间) rg_real34.13
Rg 误差 (实空间) rg_real_error1.20
I(0) (实空间) i0_real1.7000e+08
I(0) 误差 (实空间) i0_real_error2.9170e+06
Rg (倒空间) rg_reciprocal34.03
I(0) (倒空间) i0_reciprocal170000000.0000
解质量估计 total_estimate0.8361
解质量评级 solution_quality GOOD a GOOD solution
P(r) 峰数 n_peaks2
主峰位置 r_peak_primary41.1
偏度 Skewness skewness0.565
峰度 Kurtosis kurtosis0.142
角度范围 angular_range— – 0.2350 −1
当前正则化参数 α current_alpha0.0000
最高正则化参数 α highest_alpha48120000.0000
实空间数据点数 n_real_points48
GNOM 版本 gnom_version4.1.3
质量判据 quality_criteria AN1: 0.000; Oscil: 0.717; Stabil: 1.000; Sysdev: 1.000; Positv: 1.000; Valcen: 0.877; Smooth: 0.837

4. 晶体学与实验 4. Crystallography & Experiment

5. 实体与聚合体信息 (5)

6. 折叠分类 (SCOP + CATH) 11 domains

SCOP 2.08 (5 domains)

结构域编号 domain_idd1he8a1
类 Class classa — All alpha proteins
折叠类型 Fold folda.118 — alpha-alpha superhelix
超家族 Superfamily superfamilya.118.1 — ARM repeat
家族 Family familya.118.1.6 — Phoshoinositide 3-kinase (PI3K) helical domain
结构域编号 domain_idd1he8a2
类 Class classb — All beta proteins
折叠类型 Fold foldb.7 — C2 domain-like
超家族 Superfamily superfamilyb.7.1 — C2 domain (Calcium/lipid-binding domain, CaLB)
家族 Family familyb.7.1.1 — PLC-like (P variant)
结构域编号 domain_idd1he8a3
类 Class classd — Alpha and beta proteins (a+b)
折叠类型 Fold foldd.15 — beta-Grasp (ubiquitin-like)
超家族 Superfamily superfamilyd.15.1 — Ubiquitin-like
家族 Family familyd.15.1.5 — Ras-binding domain, RBD
结构域编号 domain_idd1he8a4
类 Class classd — Alpha and beta proteins (a+b)
折叠类型 Fold foldd.144 — Protein kinase-like (PK-like)
超家族 Superfamily superfamilyd.144.1 — Protein kinase-like (PK-like)
家族 Family familyd.144.1.4 — Phoshoinositide 3-kinase (PI3K), catalytic domain
结构域编号 domain_idd1he8b_
类 Class classc — Alpha and beta proteins (a/b)
折叠类型 Fold foldc.37 — P-loop containing nucleoside triphosphate hydrolases
超家族 Superfamily superfamilyc.37.1 — P-loop containing nucleoside triphosphate hydrolases
家族 Family familyc.37.1.8 — G proteins

CATH v4.4 (6 domains)

结构域编号 domain_id1he8A01
类 Class class3 — Alpha Beta
架构 Architecture architecture10 — Roll
拓扑 Topology topology20 — Ubiquitin-like (UB roll)
同源超家族 H-superfamily homologous superfamily90 — Phosphatidylinositol 3-kinase Catalytic Subunit; Chain A, domain 1
结构域编号 domain_id1he8A02
类 Class class2 — Mainly Beta
架构 Architecture architecture60 — Sandwich
拓扑 Topology topology40 — Immunoglobulin-like
同源超家族 H-superfamily homologous superfamily150 — C2 domain
结构域编号 domain_id1he8A03
类 Class class1 — Mainly Alpha
架构 Architecture architecture25 — Alpha Horseshoe
拓扑 Topology topology40 — Serine Threonine Protein Phosphatase 5, Tetratricopeptide repeat
同源超家族 H-superfamily homologous superfamily70 — Phosphatidylinositol 3-kinase, accessory domain (PIK)
结构域编号 domain_id1he8A04
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology1010 — Phosphatidylinositol 3-kinase Catalytic Subunit; Chain A, domain 4
同源超家族 H-superfamily homologous superfamily10 — Phosphatidylinositol 3-kinase Catalytic Subunit; Chain A, domain 4
结构域编号 domain_id1he8A05
类 Class class1 — Mainly Alpha
架构 Architecture architecture10 — Orthogonal Bundle
拓扑 Topology topology1070 — Phosphatidylinositol 3-kinase Catalytic Subunit; Chain A, Domain 5
同源超家族 H-superfamily homologous superfamily11 — Phosphatidylinositol 3-/4-kinase, catalytic domain
结构域编号 domain_id1he8B00
类 Class class3 — Alpha Beta
架构 Architecture architecture40 — 3-Layer(aba) Sandwich
拓扑 Topology topology50 — Rossmann fold
同源超家族 H-superfamily homologous superfamily300 — P-loop containing nucleotide triphosphate hydrolases

7. 引用文献 (1)

8. 文件与曲线 (10)