2drd

Crystal structure of a multidrug transporter reveal a functionally rotating mechanism

Method: X-RAY DIFFRACTION Dmax: 145.3 Å Quality: GOOD

SAXS 散射曲线 SAXS Profile

SAXS profile for 2drd

P(r) 距离分布 P(r) Distribution

P(r) distribution for 2drd
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1. 结构基本信息 1. Structure Basics

条目编号 entry_id2drd
沉积日期 deposition_date2006-06-08
结构标题 titleCrystal structure of a multidrug transporter reveal a functionally rotating mechanism
关键词 keywordsmembrane transporter, membrane protein, multidrug efflux, drug resistance, transporter, exporter, antiporter; MEMBRANE PROTEIN
实验方法 methodX-RAY DIFFRACTION

2. SAXS 参数 (CRYSOL 理论计算) 2. SAXS Parameters (CRYSOL)

回转半径 Rg (Guinier) rg_guinier45.45
回转半径 Rg (电子) rg_electron44.88
零角强度 I(0) i01455120000.00
分子量 molecular_weight332170.0 kDa
排除体积 excluded_volume422080 ų
包络体积 envelope_volume556150 ų
水化壳体积 shell_volume97994 ų
包络直径 envelope_diameter145.5
壳层 Rg shell_rg53.74
包络 Rg envelope_rg44.05
形状 Rg shape_rg44.89
总 Rg total_rg45.21
总原子数 total_atoms23355
残基数 n_residues3066
球谐函数阶数 n_harmonics20
q 范围 q_range— – 0.5000 −1
数据点数 n_points101
壳层类型 shell_typedirectional
溶剂电子密度 solvent_density0.3340 e/ų
壳层衬度 contrast_shell0.0300 e/ų
CRYSOL 版本 crysol_version4.1.3

3. P(r) 距离分布 (GNOM 反演) 3. P(r) Analysis (GNOM)

最大尺寸 Dmax dmax145.3
Rg (实空间) rg_real45.18
Rg 误差 (实空间) rg_real_error1.20
I(0) (实空间) i0_real1.4550e+09
I(0) 误差 (实空间) i0_real_error2.8380e+07
Rg (倒空间) rg_reciprocal45.45
I(0) (倒空间) i0_reciprocal1456000000.0000
解质量估计 total_estimate0.8853
解质量评级 solution_quality GOOD a GOOD solution
P(r) 峰数 n_peaks1
主峰位置 r_peak_primary58.1
偏度 Skewness skewness0.147
峰度 Kurtosis kurtosis-0.430
角度范围 angular_range— – 0.1750 −1
当前正则化参数 α current_alpha0.0000
最高正则化参数 α highest_alpha240200000.0000
实空间数据点数 n_real_points36
GNOM 版本 gnom_version4.1.3
质量判据 quality_criteria AN1: 0.000; Oscil: 0.868; Stabil: 1.000; Sysdev: 1.000; Positv: 1.000; Valcen: 0.981; Smooth: 0.918

4. 晶体学与实验 4. Crystallography & Experiment

5. 实体与聚合体信息 (2)

6. 折叠分类 (SCOP + CATH) 24 domains

CATH v4.4 (24 domains)

结构域编号 domain_id2drdA01
类 Class class1 — Mainly Alpha
架构 Architecture architecture20 — Up-down Bundle
拓扑 Topology topology1640 — Multidrug efflux transporter AcrB transmembrane fold
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB transmembrane domain
结构域编号 domain_id2drdA02
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1430 — Multidrug efflux transporter AcrB pore domain
结构域编号 domain_id2drdA03
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1320 — Multidrug efflux transporter AcrB pore domain like
结构域编号 domain_id2drdA04
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology2090 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
结构域编号 domain_id2drdA05
类 Class class1 — Mainly Alpha
架构 Architecture architecture20 — Up-down Bundle
拓扑 Topology topology1640 — Multidrug efflux transporter AcrB transmembrane fold
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB transmembrane domain
结构域编号 domain_id2drdA06
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1430 — Multidrug efflux transporter AcrB pore domain
结构域编号 domain_id2drdA07
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1440 — Multidrug efflux transporter AcrB pore domain
结构域编号 domain_id2drdA08
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology2090 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
结构域编号 domain_id2drdB01
类 Class class1 — Mainly Alpha
架构 Architecture architecture20 — Up-down Bundle
拓扑 Topology topology1640 — Multidrug efflux transporter AcrB transmembrane fold
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB transmembrane domain
结构域编号 domain_id2drdB02
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1430 — Multidrug efflux transporter AcrB pore domain
结构域编号 domain_id2drdB03
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1320 — Multidrug efflux transporter AcrB pore domain like
结构域编号 domain_id2drdB04
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology2090 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
结构域编号 domain_id2drdB05
类 Class class1 — Mainly Alpha
架构 Architecture architecture20 — Up-down Bundle
拓扑 Topology topology1640 — Multidrug efflux transporter AcrB transmembrane fold
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB transmembrane domain
结构域编号 domain_id2drdB06
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1430 — Multidrug efflux transporter AcrB pore domain
结构域编号 domain_id2drdB07
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1440 — Multidrug efflux transporter AcrB pore domain
结构域编号 domain_id2drdB08
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology2090 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
结构域编号 domain_id2drdC01
类 Class class1 — Mainly Alpha
架构 Architecture architecture20 — Up-down Bundle
拓扑 Topology topology1640 — Multidrug efflux transporter AcrB transmembrane fold
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB transmembrane domain
结构域编号 domain_id2drdC02
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1430 — Multidrug efflux transporter AcrB pore domain
结构域编号 domain_id2drdC03
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1320 — Multidrug efflux transporter AcrB pore domain like
结构域编号 domain_id2drdC04
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology2090 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
结构域编号 domain_id2drdC05
类 Class class1 — Mainly Alpha
架构 Architecture architecture20 — Up-down Bundle
拓扑 Topology topology1640 — Multidrug efflux transporter AcrB transmembrane fold
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB transmembrane domain
结构域编号 domain_id2drdC06
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1430 — Multidrug efflux transporter AcrB pore domain
结构域编号 domain_id2drdC07
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology70 — Alpha-Beta Plaits
同源超家族 H-superfamily homologous superfamily1440 — Multidrug efflux transporter AcrB pore domain
结构域编号 domain_id2drdC08
类 Class class3 — Alpha Beta
架构 Architecture architecture30 — 2-Layer Sandwich
拓扑 Topology topology2090 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains
同源超家族 H-superfamily homologous superfamily10 — Multidrug efflux transporter AcrB TolC docking domain; DN and DC subdomains

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