Crystal structure of human ATAD2 bromodomain in complex with N-(4-bromo-3-((3-methylpiperidin-1-yl)sulfonyl)phenyl)-2-(2,5-dioxoimidazolidin-1-yl)acetamide
Method: X-RAY DIFFRACTION
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1. 蛋白身份与相关结构 Protein Identity & Related Structures
Crystal structure of human ATAD2 bromodomain in complex with N-(4-bromo-3-((3-methylpiperidin-1-yl)sulfonyl)phenyl)-2-(2,5-dioxoimidazolidin-1-yl)acetamide
关键词 keywords
INHIBITOR, ATAD2, BROMODOMAIN, EPIGENETICS, ATPase family AAA domain-containing protein 2, transcription; TRANSCRIPTION
实验方法 method
X-RAY DIFFRACTION
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3. Official assembly/model 理论 SAXS Official SAXS Profiles
;A Qualified Success: Discovery of a New Series of ATAD2 Bromodomain Inhibitors with a Novel Binding Mode Using High-Throughput Screening and Hit Qualification.
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