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1c2l

RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES

Method: X-RAY DIFFRACTION Dmax: 52.9 Å Quality: GOOD

SAXS Profile

SAXS profile for 1c2l

P(r) Distribution

P(r) distribution for 1c2l

1. Structure Basics

entry_id1c2l
deposition_date1999-07-21
titleRECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
keywords;ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX ;; HYDROLASE/HYDROLASE INHIBITOR
methodX-RAY DIFFRACTION

Download Data

2. SAXS Parameters (CRYSOL)

rg_guinier17.09
rg_electron16.03
i010839100.00
molecular_weight23518.0 kDa
excluded_volume28982 ų
envelope_volume31755 ų
shell_volume16357 ų
envelope_diameter54.1
shell_rg22.33
envelope_rg16.27
shape_rg16.04
total_rg16.96
total_atoms3223
n_residues223
n_harmonics20
q_range— – 0.5000 −1
n_points101
shell_typedirectional
solvent_density0.3340 e/ų
contrast_shell0.0300 e/ų
crysol_version4.1.3

3. P(r) Analysis (GNOM)

dmax52.9
rg_real16.97
rg_real_error0.22
i0_real1.0840e+07
i0_real_error1.1230e+05
rg_reciprocal16.99
i0_reciprocal10840000.0000
total_estimate0.8981
solution_quality GOOD a GOOD solution
n_peaks2
r_peak_primary22.3
skewness0.124
kurtosis-0.451
angular_range— – 0.4650 −1
current_alpha0.0000
highest_alpha2815000.0000
n_real_points77
gnom_version4.1.3
quality_criteria AN1: 0.000; Oscil: 0.901; Stabil: 1.000; Sysdev: 1.000; Positv: 1.000; Valcen: 0.989; Smooth: 0.981

4. Crystallography & Experiment

5. Entities & Polymer Info (5)

6. Citations (1)

7. Files & Curves (10)